DOI: 10.1021/jm970205r. Discovery of Potent Nonpeptide Vitronectin Receptor (α<sub>V</sub>β<sub>3</sub>) Antagonists

Discovery of Potent Nonpeptide Vitronectin Receptor (αVβ3) Antagonists

10.1021/jm970205r

Crossref journal-article

American Chemical Society (ACS)

Journal of Medicinal Chemistry (316)

Bibliography

Keenan, R. M., Miller, W. H., Kwon, C., Ali, F. E., Callahan, J. F., Calvo, R. R., Hwang, S.-M., Kopple, K. D., Peishoff, C. E., Samanen, J. M., Wong, A. S., Yuan, C.-K., & Huffman, W. F. (1997). Discovery of Potent Nonpeptide Vitronectin Receptor (Î±VÎ²3) Antagonists. Journal of Medicinal Chemistry, 40(15), 2289â2292.

Authors 13

Richard M. Keenan (first)
William H. Miller (additional)
Chet Kwon (additional)
Fadia E. Ali (additional)
James F. Callahan (additional)
Raul R. Calvo (additional)
Shing-Mei Hwang (additional)
Kenneth D. Kopple (additional)
Catherine E. Peishoff (additional)
James M. Samanen (additional)
Angela S. Wong (additional)
Chuan-Kui Yuan (additional)
William F. Huffman (additional)

References 29 Referenced 103

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10.1016/S0021-9258(18)47235-3 / J. Biol. Chem. by Loftus J. C. (1994)
10.1002/jbmr.5650090709 / J. Bone Mineral Res. by Van der Pluijm G. (1994)
{'key': 'jm970205rb00002/jm970205rb00002_2', 'first-page': '343', 'volume': '7', 'author': 'Helfrich M. H.', 'year': '1992', 'journal-title': 'J. Bone Mineral Res.'} / J. Bone Mineral Res. by Helfrich M. H. (1992)
10.1016/0014-4827(91)90386-9 / Exp. Cell Res. by Horton M. A. (1991)
{'key': 'jm970205rb00003/jm970205rb00003_1', 'first-page': '134', 'volume': '19', 'author': 'Choi E. T.', 'year': '1994', 'journal-title': 'J. Vasc. Surgery'} / J. Vasc. Surgery by Choi E. T. (1994)
10.1161/01.CIR.90.5.2203 / Circulation by Matsuno H. (1994)
10.1126/science.7512751 / Science by Brooks P. C. (1994)
10.1016/0092-8674(94)90007-8 / Cell by Brooks P. C. (1994)
{'key': 'jm970205rb00005/jm970205rb00005_1', 'first-page': '533', 'volume': '2', 'author': 'Hammes H.-P.', 'year': '1996', 'journal-title': 'Nature Med.'} / Nature Med. by Hammes H.-P. (1996)
10.1073/pnas.93.18.9764 / Proc. Natl. Acad. Sci. U.S.A. by Friedlander M. (1996)
{'key': 'jm970205rb00006/jm970205rb00006_1', 'first-page': '3111', 'volume': '56', 'author': 'Yun Z.', 'year': '1996', 'journal-title': 'Cancer Res.'} / Cancer Res. by Yun Z. (1996)
{'key': 'jm970205rb00007/jm970205rb00007_1', 'first-page': '237', 'volume-title': 'I.', 'author': 'For', 'year': '1995'} / I. by For (1995)
10.1021/jm00099a026 / J. Med. Chem. by Peishoff C. E. (1992)
10.1021/jm00099a027 / J. Med. Chem. by Callahan J. F. (1992)
{'key': 'jm970205rb00010/jm970205rb00010_1', 'first-page': '780', 'volume': '37', 'author': 'Ali F. E.', 'year': '1994', 'journal-title': 'J. Med. Chem.'} / J. Med. Chem. by Ali F. E. (1994)
{'key': 'jm970205rb00011/jm970205rb00011_1', 'first-page': '8862', 'volume': '115', 'author': 'Ku T. W.', 'year': '1993', 'journal-title': 'J. Am. Chem. Soc.'} / J. Am. Chem. Soc. by Ku T. W. (1993)
10.1016/S0968-0896(00)82039-8 / Bioorg. Med. Chem. by Bondinell W. E. (1994)
{'key': 'jm970205rb00013/jm970205rb00013_1', 'first-page': '12', 'volume': '38', 'author': 'Ku T. W.', 'year': '1995', 'journal-title': 'J. Med. Chem.'} / J. Med. Chem. by Ku T. W. (1995)
10.1021/jm960558a / J. Med. Chem. by Samanen J. M. (1996)
{'key': 'jm970205rb00015/jm970205rb00015_1', 'first-page': '921', 'volume': '292', 'author': 'Gurrath M.', 'year': '1992', 'journal-title': 'FEBS'} / FEBS by Gurrath M. (1992)
10.1016/0014-5793(91)81101-D / FEBS Lett. by Aumailley M. (1991)
{'key': 'jm970205rb00016/jm970205rb00016_1', 'volume-title': 'A.', 'author': 'Binding SK', 'year': '1996'} / A. by Binding SK (1996)
Ali, F. E.; Samanen, J. M.; Synthesis of Protected Cyclic Homodetic Peptides by Solid Phase Peptide Synthesis. InInnovations and Perspectives in Solid Phase Synthesis & Related Technologies; Epton, R., Ed.; SPCC (UK) Ltd. London, 1991; pp 333−335.
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{'key': 'jm970205rb00021/jm970205rb00021_1', 'first-page': 'S288', 'volume': '11', 'author': 'James I. E.', 'year': '1996', 'journal-title': 'J. Bone Mineral Res.'} / J. Bone Mineral Res. by James I. E. (1996)
10.1159/000159159 / J. Vascular Res. by Powers D. A. (1996)
A preliminary account of this work was presented at the 211th American Chemical Society National Meeting, New Orleans, LA, March 24−28, 1996.

Dates

Type	When
Created	23 years, 1 month ago (July 26, 2002, 1:10 a.m.)
Deposited	1 year, 7 months ago (Jan. 2, 2024, 5:52 p.m.)
Indexed	3 months ago (May 22, 2025, 3:11 a.m.)
Issued	28 years, 1 month ago (July 1, 1997)
Published	28 years, 1 month ago (July 1, 1997)
Published Online	28 years, 1 month ago (July 18, 1997)
Published Print	28 years, 1 month ago (July 1, 1997)

Funders 0

None

BibTeX

@article{Keenan_1997, title={Discovery of Potent Nonpeptide Vitronectin Receptor (αVβ3) Antagonists}, volume={40}, ISSN={1520-4804}, url={http://dx.doi.org/10.1021/jm970205r}, DOI={10.1021/jm970205r}, number={15}, journal={Journal of Medicinal Chemistry}, publisher={American Chemical Society (ACS)}, author={Keenan, Richard M. and Miller, William H. and Kwon, Chet and Ali, Fadia E. and Callahan, James F. and Calvo, Raul R. and Hwang, Shing-Mei and Kopple, Kenneth D. and Peishoff, Catherine E. and Samanen, James M. and Wong, Angela S. and Yuan, Chuan-Kui and Huffman, William F.}, year={1997}, month=jul, pages={2289–2292} }

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