DOI: 10.1021/jm9505167. Structure−Activity Analysis of Anandamide Analogs: Relationship to a Cannabinoid Pharmacophore

Structure−Activity Analysis of Anandamide Analogs: Relationship to a Cannabinoid Pharmacophore

10.1021/jm9505167

Crossref journal-article

American Chemical Society (ACS)

Journal of Medicinal Chemistry (316)

Bibliography

Thomas, B. F., Adams, I. B., Mascarella, S. W., Martin, B. R., & Razdan, R. K. (1996). StructureâActivity Analysis of Anandamide Analogs:â Relationship to a Cannabinoid Pharmacophore. Journal of Medicinal Chemistry, 39(2), 471â479.

Authors 5

Brian F. Thomas (first)
Irma B. Adams (additional)
S. Wayne Mascarella (additional)
Billy R. Martin (additional)
Raj K. Razdan (additional)

References 27 Referenced 61

10.1126/science.1470919 / Science by Devane W. A. (1992)
10.1111/j.1471-4159.1993.tb03576.x / J. Neurochem. by Vogel Z. (1993)
{'key': 'jm9505167b00003/jm9505167b00003_1', 'first-page': '7660', 'volume': '90', 'author': 'Felder C. C.', 'year': '1993', 'journal-title': 'PNAS'} / PNAS by Felder C. C. (1993)
10.1016/0014-2999(93)90468-W / Eur. J. Pharmacol. by Fride E. (1993)
{'key': 'jm9505167b00005/jm9505167b00005_1', 'first-page': '227', 'volume': '270', 'author': 'Smith P. B.', 'year': '1994', 'journal-title': 'J. Pharmacol. Exp. Ther.'} / J. Pharmacol. Exp. Ther. by Smith P. B. (1994)
{'key': 'jm9505167b00006/jm9505167b00006_1', 'first-page': '1181', 'volume': '273', 'author': 'Adams I. B.', 'year': '1995', 'journal-title': 'J. Pharmacol. Exp. Ther.'} / J. Pharmacol. Exp. Ther. by Adams I. B. (1995)
10.1016/0091-3057(93)90230-Q / Pharmacol. Biochem. Behav. by Crawley J. N. (1993)
10.1021/jm00072a026 / J. Med. Chem. by Hanus L. (1993)
{'key': 'jm9505167b00009/jm9505167b00009_1', 'first-page': '522', 'volume': '46', 'author': 'Pinto J. C.', 'year': '1994', 'journal-title': 'Mol. Pharmacol.'} / Mol. Pharmacol. by Pinto J. C. (1994)
10.1021/jm00038a020 / J. Med. Chem. by Abadji V. (1994)
{'key': 'jm9505167b00011/jm9505167b00011_1', 'first-page': '161', 'volume-title': 'Neuroreceptors', 'author': 'Binder M.', 'year': '1982'} / Neuroreceptors by Binder M. (1982)
{'key': 'jm9505167b00012/jm9505167b00012_1', 'first-page': '149', 'volume': '38', 'author': 'Razdan R. K', 'year': '1986', 'journal-title': 'Pharm. Rev.'} / Pharm. Rev. by Razdan R. K (1986)
10.1021/jm00127a038 / J. Med. Chem. by Reggio P. H. (1989)
{'key': 'jm9505167b00014/jm9505167b00014_1', 'first-page': '503', 'volume': '35', 'author': 'Kriwacki R. W.', 'year': '1989', 'journal-title': 'Mol. Pharmacol.'} / Mol. Pharmacol. by Kriwacki R. W. (1989)
{'key': 'jm9505167b00015/jm9505167b00015_1', 'first-page': '665', 'volume': '40', 'author': 'Thomas B. F.', 'year': '1991', 'journal-title': 'Mol. Pharmacol.'} / Mol. Pharmacol. by Thomas B. F. (1991)
10.1002/j.1552-4604.1981.tb02616.x / J. Clin, Pharmacol. by Milne G. M. (1981)
{'key': 'jm9505167b00017/jm9505167b00017_1', 'first-page': '145', 'volume-title': 'Cannabinoids as Therapeutic Agents', 'author': 'Johnson M. R.', 'year': '1986'} / Cannabinoids as Therapeutic Agents by Johnson M. R. (1986)
{'key': 'jm9505167b00018/jm9505167b00018_1', 'first-page': '613', 'volume': '34', 'author': 'Devane W. A.', 'year': '1988', 'journal-title': 'Mol. Pharmacol.'} / Mol. Pharmacol. by Devane W. A. (1988)
{'key': 'jm9505167b00019/jm9505167b00019_1', 'first-page': '96', 'volume': '1178', 'author': 'Rich M. R', 'year': '1993', 'journal-title': 'Biochim. Biophys. Acta'} / Biochim. Biophys. Acta by Rich M. R (1993)
10.1021/ja00500a036 / J. Am. Chem. Soc. by Corey E. J. (1979)
10.1016/S0040-4039(00)81320-9 / Tetrahedron Lett. by Corey E. J. (1983)
{'key': 'jm9505167b00022/jm9505167b00022_1', 'first-page': '228', 'volume': '134', 'author': 'Reggio P. H', 'year': '1993', 'journal-title': 'Natl. Inst. Drug Abuse Res. Monogr.'} / Natl. Inst. Drug Abuse Res. Monogr. by Reggio P. H (1993)
Thibaut, U.; Folkers, G.; Klebe, G.; Kubinyi, H.; Merz, A.; Rognan, D. Recommendations for CoMFA Studies and 3D QSAR Publications. In3D QSAR in Drug Design: Theory,Methods and Applications; Kubinyi, H., Ed., ESCOM: Leiden, 1993; pp 711−716. (10.1002/qsar.19940130102)
10.1021/jm00367a013 / J. Med. Chem. by Melvin L. S. (1984)
{'key': 'jm9505167b00025/jm9505167b00025_1', 'first-page': '95', 'volume': '79', 'author': 'Reggio P. H', 'year': '1987', 'journal-title': 'Natl. Inst. Drug Abuse Res. Monogr.'} / Natl. Inst. Drug Abuse Res. Monogr. by Reggio P. H (1987)
10.1016/S0960-894X(01)80155-4 / Biomed. Chem. Lett. by Huffman J. W. (1994)
{'key': 'jm9505167b00027/jm9505167b00027_1', 'first-page': '1015', 'volume': '44', 'author': 'Melvin L. S.', 'year': '1993', 'journal-title': 'Mol. Pharmacol.'} / Mol. Pharmacol. by Melvin L. S. (1993)

Dates

Type	When
Created	23 years, 1 month ago (July 26, 2002, 2 a.m.)
Deposited	3 years, 11 months ago (Sept. 22, 2021, 11:52 p.m.)
Indexed	11 months, 3 weeks ago (Sept. 10, 2024, 3:51 p.m.)
Issued	29 years, 8 months ago (Jan. 1, 1996)
Published	29 years, 8 months ago (Jan. 1, 1996)
Published Online	29 years, 7 months ago (Jan. 19, 1996)
Published Print	29 years, 8 months ago (Jan. 1, 1996)

Funders 0

None

BibTeX

@article{Thomas_1996, title={Structure‚àíActivity Analysis of Anandamide Analogs:‚Äâ Relationship to a Cannabinoid Pharmacophore}, volume={39}, ISSN={1520-4804}, url={http://dx.doi.org/10.1021/jm9505167}, DOI={10.1021/jm9505167}, number={2}, journal={Journal of Medicinal Chemistry}, publisher={American Chemical Society (ACS)}, author={Thomas, Brian F. and Adams, Irma B. and Mascarella, S. Wayne and Martin, Billy R. and Razdan, Raj K.}, year={1996}, month=jan, pages={471‚Äì479} }

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