DOI: 10.1021/ja034247i. Discovery of a Potent Small Molecule IL-2 Inhibitor through Fragment Assembly

Discovery of a Potent Small Molecule IL-2 Inhibitor through Fragment Assembly

10.1021/ja034247i

Crossref journal-article

American Chemical Society (ACS)

Journal of the American Chemical Society (316)

Bibliography

Braisted, A. C., Oslob, J. D., Delano, W. L., Hyde, J., McDowell, R. S., Waal, N., Yu, C., Arkin, M. R., & Raimundo, B. C. (2003). Discovery of a Potent Small Molecule IL-2 Inhibitor through Fragment Assembly. Journal of the American Chemical Society, 125(13), 3714â3715.

Authors 9

Andrew C. Braisted (first)
Johan D. Oslob (additional)
Warren L. Delano (additional)
Jennifer Hyde (additional)
Robert S. McDowell (additional)
Nathan Waal (additional)
Chul Yu (additional)
Michelle R. Arkin (additional)
Brian C. Raimundo (additional)

References 12 Referenced 218

10.1021/jm010468s / J. Med. Chem. by Toogood P. L. (2002)
10.1016/S1367-5931(01)00262-9 / Curr. Opin. Chem. Biol. by Cochran A. G. (2001)
10.1021/cr960387h / Chem. Rev. by Stites W. E. (1997)
10.1126/science.274.5292.1531 / Science by Shuker S. B. (1996)
10.1038/nrd704 / Nat. Rev. Drug Discovery by Ramstrom O. (2002)
10.1016/S1367-5931(02)00331-9 / Curr. Opin. Chem. Biol. by Otto S. (2002)
10.1021/jm000017s / J. Med. Chem. by Boehm H. J. (2000)
10.1073/pnas.97.17.9367 / Proc. Natl. Acad. Sci. U.S.A. by Erlanson D. A. (2000)
{'key': 'ja034247ib00004/ja034247ib00004_1', 'first-page': '81', 'volume': '70', 'author': 'Nelson B. H.', 'year': '1998', 'journal-title': 'Adv. Immunol.'} / Adv. Immunol. by Nelson B. H. (1998)
10.1021/ja970702x / J. Am. Chem. Soc. by Tilley J. W. (1997)
Raimundo, B. C.; Oslob, J. D.; Hyde, J.; Randal, M.; Waal, N.; Yu, C.; Arkin, M. R.2003, manuscript in preparation.
10.1073/pnas.252756299 / Proc. Natl. Acad. Sci. U.S.A. by Arkin M. R. (2003)

Dates

Type	When
Created	22 years, 5 months ago (March 26, 2003, 2:39 a.m.)
Deposited	3 years, 10 months ago (Oct. 18, 2021, 4:54 a.m.)
Indexed	1 week ago (Aug. 29, 2025, 5:59 a.m.)
Issued	22 years, 5 months ago (March 11, 2003)
Published	22 years, 5 months ago (March 11, 2003)
Published Online	22 years, 5 months ago (March 11, 2003)
Published Print	22 years, 5 months ago (April 1, 2003)

Funders 0

None

BibTeX

@article{Braisted_2003, title={Discovery of a Potent Small Molecule IL-2 Inhibitor through Fragment Assembly}, volume={125}, ISSN={1520-5126}, url={http://dx.doi.org/10.1021/ja034247i}, DOI={10.1021/ja034247i}, number={13}, journal={Journal of the American Chemical Society}, publisher={American Chemical Society (ACS)}, author={Braisted, Andrew C. and Oslob, Johan D. and Delano, Warren L. and Hyde, Jennifer and McDowell, Robert S. and Waal, Nathan and Yu, Chul and Arkin, Michelle R. and Raimundo, Brian C.}, year={2003}, month=mar, pages={3714–3715} }

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