DOI: 10.1021/cg034058b. High-Throughput Surveys of Crystal Form Diversity of Highly Polymorphic Pharmaceutical Compounds

High-Throughput Surveys of Crystal Form Diversity of Highly Polymorphic Pharmaceutical Compounds

10.1021/cg034058b

Crossref journal-article

American Chemical Society (ACS)

Crystal Growth & Design (316)

Bibliography

Almarsson, Ã., Hickey, M. B., Peterson, M. L., Morissette, S. L., Soukasene, S., McNulty, C., Tawa, M., MacPhee, J. M., & Remenar, J. F. (2003). High-Throughput Surveys of Crystal Form Diversity of Highly Polymorphic Pharmaceutical Compounds. Crystal Growth & Design, 3(6), 927â933.

Authors 9

Örn Almarsson (first)
Magali B. Hickey (additional)
Matthew L. Peterson (additional)
Sherry L. Morissette (additional)
Stephen Soukasene (additional)
Chris McNulty (additional)
Mark Tawa (additional)
J. Michael MacPhee (additional)
Julius F. Remenar (additional)

References 16 Referenced 73

{'key': 'cg034058bb00001/cg034058bb00001_1', 'volume-title': 'Polymorphism in Molecular Crystals', 'author': 'Bernstein J.', 'year': '2002'} / Polymorphism in Molecular Crystals by Bernstein J. (2002)
McCrone, W. C. inPhysics and Chemistry of the Organic Solid State; Fox, D., Labes, M. M., Weissberger, A., Eds.; Wiley-Interscience: New York, 1965; Vol. 2, pp 725−767.
{'key': 'cg034058bb00003/cg034058bb00003_1', 'volume-title': 'in Polymorphism in Pharmaceutical Solids', 'volume': '1999', 'author': 'Grant D. J. W.'} / in Polymorphism in Pharmaceutical Solids by Grant D. J. W.
(b) Byrn, S. R.; Pfeiffer, R. R.; Stowell, J. G.Solid-State Chemistry of Drugs, 2nd ed.; SSCI Inc. West Lafayette, IN, 1999; Chapter 10, p 233.
{'key': 'cg034058bb00004/cg034058bb00004_1', 'volume-title': 'MicroMedex (Thomson Healthcare)', 'author': "Physician's Desk Reference", 'year': '2003'} / MicroMedex (Thomson Healthcare) by Physician's Desk Reference (2003)
10.1023/A:1011052932607 / Pharm. Res. by Bauer J. (2001)
10.1021/op000023y / Org. Proc. Res. Dev. by Chemburkar S. R. (2000)
10.1073/pnas.0437744100 / Proc. Natl. Acad. Sci. U.S.A. by Morissette S. L. (2003)
{'key': 'cg034058bb00007/cg034058bb00007_1', 'first-page': '208', 'volume': '198', 'author': 'Caira M. R.', 'year': '1998', 'journal-title': 'Crystalline Polymorphism of Organic Compounds in Top. Curr. Chem.'} / Crystalline Polymorphism of Organic Compounds in Top. Curr. Chem. by Caira M. R. (1998)
{'key': 'cg034058bb00008/cg034058bb00008_1', 'first-page': '10959', 'volume': '124', 'author': 'Peterson M. L.', 'year': '2002', 'journal-title': 'J. Am. Chem. Soc.'} / J. Am. Chem. Soc. by Peterson M. L. (2002)
{'key': 'cg034058bb00009/cg034058bb00009_1', 'first-page': '187', 'volume': '4', 'author': 'Jahansouz H.', 'year': '1999', 'journal-title': 'J. Pharm. Dev. Technol.'} / J. Pharm. Dev. Technol. by Jahansouz H. (1999)
Phenobarbital has 13 polymorphs reported; see Kuhnert-BrandstätterThermomicroscopy in the Analysis of Pharmaceuticals; Pergamon Press: Oxford, 1971.
{'key': 'cg034058bb00012/cg034058bb00012_1', 'volume-title': 'Proceedings of the Fourth International Conference on Foundations of Computer-Aided Process Operations, Grossmann, I. E., McDonald, C. M., Eds.', 'author': 'Gardner C. R.', 'year': '2003'} / Proceedings of the Fourth International Conference on Foundations of Computer-Aided Process Operations, Grossmann, I. E., McDonald, C. M., Eds. by Gardner C. R. (2003)
10.1016/0378-5173(95)04466-3 / Int. J. Pharm. by Zhu H. (1996)
10.1021/ar00052a005 / Acc. Chem. Res. by Dunitz J. D. (1995)
{'key': 'cg034058bb00018/cg034058bb00018_1', 'volume-title': '“tailor-made', 'author': 'The'} / “tailor-made by The

Dates

Type	When
Created	21 years, 9 months ago (Nov. 5, 2003, 8:39 a.m.)
Deposited	2 years, 5 months ago (March 20, 2023, 2:37 p.m.)
Indexed	3 weeks, 6 days ago (July 25, 2025, 6:41 a.m.)
Issued	21 years, 11 months ago (Sept. 10, 2003)
Published	21 years, 11 months ago (Sept. 10, 2003)
Published Online	21 years, 11 months ago (Sept. 10, 2003)
Published Print	21 years, 9 months ago (Nov. 1, 2003)

Funders 0

None

BibTeX

@article{Almarsson_2003, title={High-Throughput Surveys of Crystal Form Diversity of Highly Polymorphic Pharmaceutical Compounds}, volume={3}, ISSN={1528-7505}, url={http://dx.doi.org/10.1021/cg034058b}, DOI={10.1021/cg034058b}, number={6}, journal={Crystal Growth & Design}, publisher={American Chemical Society (ACS)}, author={Almarsson, Örn and Hickey, Magali B. and Peterson, Matthew L. and Morissette, Sherry L. and Soukasene, Stephen and McNulty, Chris and Tawa, Mark and MacPhee, J. Michael and Remenar, Julius F.}, year={2003}, month=sep, pages={927–933} }

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