DOI: 10.1021/bi971711l. Comparison of Two Independent Crystal Structures of Human Dihydrofolate Reductase Ternary Complexes Reduced with Nicotinamide Adenine Dinucleotide Phosphate and the Very Tight-Binding Inhibitor PT523<sup>,</sup>

Comparison of Two Independent Crystal Structures of Human Dihydrofolate Reductase Ternary Complexes Reduced with Nicotinamide Adenine Dinucleotide Phosphate and the Very Tight-Binding Inhibitor PT523,

10.1021/bi971711l

Crossref journal-article

American Chemical Society (ACS)

Biochemistry (316)

Bibliography

Cody, V., Galitsky, N., Luft, J. R., Pangborn, W., Rosowsky, A., & Blakley, R. L. (1997). Comparison of Two Independent Crystal Structures of Human Dihydrofolate Reductase Ternary Complexes Reduced with Nicotinamide Adenine Dinucleotide Phosphate and the Very Tight-Binding Inhibitor PT523,. Biochemistry, 36(45), 13897â13903.

Authors 6

Vivian Cody (first)
Nikolai Galitsky (additional)
Joseph R. Luft (additional)
Walter Pangborn (additional)
Andre Rosowsky (additional)
Raymond L. Blakley (additional)

References 31 Referenced 47

{'key': 'bi971711lb00001/bi971711lb00001_1', 'volume-title': 'Folates and Pteridines', 'volume': '1', 'author': 'Blakley R. L.', 'year': '1984'} / Folates and Pteridines by Blakley R. L. (1984)
{'key': 'bi971711lb00002/bi971711lb00002_1', 'first-page': '252', 'volume': '26', 'author': 'Rosowsky A.', 'year': '1989', 'journal-title': 'Prog. Med. Chem.'} / Prog. Med. Chem. by Rosowsky A. (1989)
Blakley, R. L. (1995)Advances in Enzymology and Related Areas of Molecular Biology(Meister, A., Ed.) Vol. 70, pp 23−102, John Wiley & Sons, Inc., New York. (10.1002/9780470123164.ch2)
10.1002/j.1552-4604.1990.tb03596.x / J. Clin. Pharmacol. by Bertino J. R. (1990)
{'key': 'bi971711lb00005/bi971711lb00005_1', 'volume': '27', 'author': 'Rosowsky A.', 'year': '1984', 'journal-title': 'J. Med. Chem.'} / J. Med. Chem. by Rosowsky A. (1984)
{'key': 'bi971711lb00006/bi971711lb00006_1', 'volume': '29', 'author': 'Rosowsky A.', 'year': '1986', 'journal-title': 'J. Med. Chem.'} / J. Med. Chem. by Rosowsky A. (1986)
{'key': 'bi971711lb00007/bi971711lb00007_1', 'volume-title': 'Biochem. Pharmacol. 35, 3327−3333', 'author': 'Rosowsky A.', 'year': '1986'} / Biochem. Pharmacol. 35, 3327−3333 by Rosowsky A. (1986)
{'key': 'bi971711lb00008/bi971711lb00008_1', 'volume-title': 'Cancer Res. 50, 1720−1731', 'author': 'McGuire J. J.', 'year': '1990'} / Cancer Res. 50, 1720−1731 by McGuire J. J. (1990)
{'key': 'bi971711lb00009/bi971711lb00009_1', 'volume': '31', 'author': 'Rosowsky A.', 'year': '1988', 'journal-title': 'J. Med. Chem.'} / J. Med. Chem. by Rosowsky A. (1988)
{'key': 'bi971711lb00010/bi971711lb00010_1', 'volume-title': 'Mol. Pharmacol. 45, 783−791', 'author': 'Rhee M. S.', 'year': '1994'} / Mol. Pharmacol. 45, 783−791 by Rhee M. S. (1994)
{'key': 'bi971711lb00011/bi971711lb00011_1', 'volume-title': 'Mol. Pharmacol. 48, 758−765', 'author': 'Chen G.', 'year': '1995'} / Mol. Pharmacol. 48, 758−765 by Chen G. (1995)
{'key': 'bi971711lb00012/bi971711lb00012_1', 'volume-title': 'Mol. Pharmacol. 48, 459−471', 'author': 'Westerhof G. R.', 'year': '1995'} / Mol. Pharmacol. 48, 459−471 by Westerhof G. R. (1995)
{'key': 'bi971711lb00013/bi971711lb00013_1', 'volume-title': 'Biochemistry 36, 4399−4411', 'author': 'Johnson J. M.', 'year': '1997'} / Biochemistry 36, 4399−4411 by Johnson J. M. (1997)
{'key': 'bi971711lb00014/bi971711lb00014_1', 'volume': '34', 'author': 'Rosowsky A.', 'year': '1991', 'journal-title': 'J. Med. Chem.'} / J. Med. Chem. by Rosowsky A. (1991)
{'key': 'bi971711lb00015/bi971711lb00015_1', 'volume': '37', 'author': 'Rosowsky A.', 'year': '1994', 'journal-title': 'J. Med. Chem.'} / J. Med. Chem. by Rosowsky A. (1994)
{'key': 'bi971711lb00016/bi971711lb00016_1', 'volume': '40', 'author': 'Rosowsky A.', 'year': '1997', 'journal-title': 'J. Med. Chem.'} / J. Med. Chem. by Rosowsky A. (1997)
10.1016/S0021-9258(17)36916-8 / J. Biol. Chem. by Chunduru S. K. (1994)
{'key': 'bi971711lb00018/bi971711lb00018_1', 'volume-title': 'Anticancer Drug Des. 7, 483−491', 'author': 'Cody V.', 'year': '1992'} / Anticancer Drug Des. 7, 483−491 by Cody V. (1992)
{'key': 'bi971711lb00019/bi971711lb00019_1', 'volume-title': 'Chemistry and Biology of Pteridines and Folates', 'author': 'Cody V.', 'year': '1993'} / Chemistry and Biology of Pteridines and Folates by Cody V. (1993)
{'key': 'bi971711lb00020/bi971711lb00020_1', 'volume': '270', 'author': 'Lewis W. S.', 'year': '1995', 'journal-title': 'J. Biol. Chem.'} / J. Biol. Chem. by Lewis W. S. (1995)
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{'key': 'bi971711lb00022/bi971711lb00022_1', 'volume-title': 'Biochemistry 29, 9467−9479', 'author': 'Davies J. F.', 'year': '1990'} / Biochemistry 29, 9467−9479 by Davies J. F. (1990)
{'key': 'bi971711lb00023/bi971711lb00023_1', 'volume-title': 'XPLOR', 'author': 'Brunger A. T.', 'year': '1992'} / XPLOR by Brunger A. T. (1992)
{'key': 'bi971711lb00024/bi971711lb00024_1', 'volume-title': 'in Computing in Crystallography', 'author': 'Hendrickson W. A.', 'year': '1980'} / in Computing in Crystallography by Hendrickson W. A. (1980)
{'key': 'bi971711lb00025/bi971711lb00025_1', 'volume': '6', 'author': 'Sack J. S.', 'year': '1988', 'journal-title': 'J. Mol. Graphics'} / J. Mol. Graphics by Sack J. S. (1988)
10.1107/S0021889892009944 / J. Appl. Crystallogr. by Laskowski R. A. (1993)
10.1016/S0021-9258(18)33497-5 / J. Biol. Chem. by Bolin J. T. (1982)
10.1016/S0021-9258(18)33498-7 / J. Biol. Chem. by Filman D. S. (1982)
Kraut, J., and Matthews, D. A. (1987) inBiological Macromolecules and Assemblies(Jurnak, F., and McPherson, A., Eds.) Vol. III, pp 1−71, John Wiley and Sons: New York.
{'key': 'bi971711lb00031/bi971711lb00031_1', 'first-page': '102', 'volume': '11', 'author': 'Rossmann M. G.', 'year': '1975', 'journal-title': 'Enzymes'} / Enzymes by Rossmann M. G. (1975)
{'key': 'bi971711lb00032/bi971711lb00032_1', 'volume': '11', 'author': 'Evans S. V.', 'year': '1993', 'journal-title': 'SETOR, J. Mol. Graphics'} / SETOR, J. Mol. Graphics by Evans S. V. (1993)

Dates

Type	When
Created	23 years, 1 month ago (July 26, 2002, 1:05 a.m.)
Deposited	1 year, 7 months ago (Jan. 2, 2024, 5:08 p.m.)
Indexed	2 months, 3 weeks ago (June 6, 2025, 5:08 a.m.)
Issued	27 years, 9 months ago (Nov. 1, 1997)
Published	27 years, 9 months ago (Nov. 1, 1997)
Published Online	27 years, 9 months ago (Nov. 11, 1997)
Published Print	27 years, 9 months ago (Nov. 1, 1997)

Funders 0

None

BibTeX

@article{Cody_1997, title={Comparison of Two Independent Crystal Structures of Human Dihydrofolate Reductase Ternary Complexes Reduced with Nicotinamide Adenine Dinucleotide Phosphate and the Very Tight-Binding Inhibitor PT523,}, volume={36}, ISSN={1520-4995}, url={http://dx.doi.org/10.1021/bi971711l}, DOI={10.1021/bi971711l}, number={45}, journal={Biochemistry}, publisher={American Chemical Society (ACS)}, author={Cody, Vivian and Galitsky, Nikolai and Luft, Joseph R. and Pangborn, Walter and Rosowsky, Andre and Blakley, Raymond L.}, year={1997}, month=nov, pages={13897–13903} }

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