DOI: 10.1021/bi00047a010. .alpha.-Fluoro Acid and .alpha.-Fluoro Amide Analogs of Acetyl-CoA as Inhibitors of Citrate Synthase: Effect of pKa Matching on Binding Affinity and Hydrogen Bond Length

.alpha.-Fluoro Acid and .alpha.-Fluoro Amide Analogs of Acetyl-CoA as Inhibitors of Citrate Synthase: Effect of pKa Matching on Binding Affinity and Hydrogen Bond Length

10.1021/bi00047a010

Crossref journal-article

American Chemical Society (ACS)

Biochemistry (316)

Bibliography

Schwartz, B., Drueckhammer, D. G., Usher, K. C., & Remington, S. J. (1995). .alpha.-Fluoro Acid and .alpha.-Fluoro Amide Analogs of Acetyl-CoA as Inhibitors of Citrate Synthase: Effect of pKa Matching on Binding Affinity and Hydrogen Bond Length. Biochemistry, 34(47), 15459â15466.

Authors 4

Benjamin Schwartz (first)
Dale G. Drueckhammer (additional)
Ken C. Usher (additional)
S. James Remington (additional)

References 0 Referenced 29

None

Dates

Type	When
Created	20 years, 5 months ago (March 8, 2005, 6:19 a.m.)
Deposited	2 years, 5 months ago (March 7, 2023, 5:27 a.m.)
Indexed	1 year, 7 months ago (Jan. 12, 2024, 6 p.m.)
Issued	29 years, 10 months ago (Nov. 1, 1995)
Published	29 years, 10 months ago (Nov. 1, 1995)
Published Online	23 years, 4 months ago (May 1, 2002)
Published Print	29 years, 10 months ago (Nov. 1, 1995)

Funders 0

None

BibTeX

@article{Schwartz_1995, title={.alpha.-Fluoro Acid and .alpha.-Fluoro Amide Analogs of Acetyl-CoA as Inhibitors of Citrate Synthase: Effect of pKa Matching on Binding Affinity and Hydrogen Bond Length}, volume={34}, ISSN={1520-4995}, url={http://dx.doi.org/10.1021/bi00047a010}, DOI={10.1021/bi00047a010}, number={47}, journal={Biochemistry}, publisher={American Chemical Society (ACS)}, author={Schwartz, Benjamin and Drueckhammer, Dale G. and Usher, Ken C. and Remington, S. James}, year={1995}, month=nov, pages={15459–15466} }

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