Bibliography
Zhang, D., Saraf, A., Kolasa, T., Bhatia, P., Zheng, G. Z., Patel, M., Lannoye, G. S., Richardson, P., Stewart, A., Rogers, J. C., Brioni, J. D., & Surowy, C. S. (2007). Fatty acid amide hydrolase inhibitors display broad selectivity and inhibit multiple carboxylesterases as off-targets. Neuropharmacology, 52(4), 1095â1105.
Authors
12
- Di Zhang (first)
- Anita Saraf (additional)
- Teodozyi Kolasa (additional)
- Pramila Bhatia (additional)
- Guo Zhu Zheng (additional)
- Meena Patel (additional)
- Greg S. Lannoye (additional)
- Paul Richardson (additional)
- Andrew Stewart (additional)
- John C. Rogers (additional)
- Jorge D. Brioni (additional)
- Carol S. Surowy (additional)
References
47
Referenced
86
- Abouabdellah, A., Bas, M., Dargazanli, G., Hoornaert, C., Li, A.T., Medaisko, F., 2005. Derivatives of dioxane-2-alkyl carbamates, preparation thereof and application thereof in therapeutics. Patent US20050182130 A1.
- Abouabdellah, A., Burnier, P., Hoornaert, C., Jeunesse, J., Puech, F., 2006. Derivatives of piperidinyl- and piperazinyl-alkyl carbamates, preparation methods thereof and application of some in therapeutics. Patent US20060089344 A1.
10.1016/j.chembiol.2005.08.011
/ Chem. Biol. / Mechanism of carbamate inactivation of FAAH: implications for the design of covalent inhibitors and in vivo functional probes for enzymes by Alexander (2005)10.1021/ja062999h
/ J. Am. Chem. Soc. / The putative endocannabinoid transport blocker LY2183240 is a potent inhibitor of FAAH and several other brain serine hydrolases by Alexander (2006)10.1161/01.CIR.0000143230.23252.D2
/ Circulation / Endocannabinoids acting at cannabinoid-1 receptors regulate cardiovascular function in hypertension by Batkai (2004)10.1126/science.277.5329.1094
/ Science / Functional role of high-affinity anandamide transport, as revealed by selective inhibition by Beltramo (1997)- Boger, D.L., 2004. Inhibitors of fatty acid amide hydrolase. Patent WO2004033652 A2.
10.1021/jm049614v
/ J. Med. Chem. / Discovery of a potent, selective, and efficacious class of reversible alpha-ketoheterocycle inhibitors of fatty acid amide hydrolase effective as analgesics by Boger (2005)10.1073/pnas.97.10.5044
/ Proc. Natl. Acad. Sci. U.S.A. / Exceptionally potent inhibitors of fatty acid amide hydrolase: the enzyme responsible for degradation of endogenous oleamide and anandamide by Boger (2000)10.1126/science.1076535
/ Science / Structural adaptations in a membrane enzyme that terminates endocannabinoid signaling by Bracey (2002)10.1016/S0014-2999(97)01297-1
/ Eur. J. Pharmacol. / Potentiation of anandamide hypotension by the transport inhibitor, AM404 by Calignano (1997)10.1038/sj.bjp.0706699
/ Br. J. Pharmacol. / Inhibition of fatty acid amide hydrolase produces analgesia by multiple mechanisms by Chang (2006)10.1016/j.phrs.2006.06.008
/ Pharmacol. Res. / The fatty-acid amide hydrolase inhibitor URB597 does not affect triacylglycerol hydrolysis in rat tissues by Clapper (2006)10.1073/pnas.161191698
/ Proc. Natl. Acad. Sci. U.S.A. / Supersensitivity to anandamide and enhanced endogenous cannabinoid signaling in mice lacking fatty acid amide hydrolase by Cravatt (2001)10.1016/S1367-5931(03)00079-6
/ Curr. Opin. Chem. Biol. / Fatty acid amide hydrolase: an emerging therapeutic target in the endocannabinoid system by Cravatt (2003)10.1054/plef.2001.0349
/ Prostaglandins Leukot. Essent. Fatty Acids / Anandamide receptors by Di Marzo (2002)10.1007/s00018-004-3426-3
/ Cell. Mol. Life Sci. / Triacylglycerol hydrolase: role in intracellular lipid metabolism by Dolinsky (2004)10.1016/j.bcp.2005.01.017
/ Biochem. Pharmacol. / Dexamethasone-induced methylprednisolone hemisuccinate hydrolase: its identification as a member of the rat carboxylesterase 2 family and its unique existence in plasma by Furihata (2005)10.1073/pnas.0730816100
/ Proc. Natl. Acad. Sci. U.S.A. / Evidence against the presence of an anandamide transporter by Glaser (2003)10.1073/pnas.0509591102
/ Proc. Natl. Acad. Sci. U.S.A. / Antidepressant-like activity and modulation of brain monoaminergic transmission by blockade of anandamide hydrolysis by Gobbi (2005)10.1038/sj.bjp.0706348
/ Br. J. Pharmacol. / Inhibitors of fatty acid amide hydrolase reduce carrageenan-induced hind paw inflammation in pentobarbital-treated mice: comparison with indomethacin and possible involvement of cannabinoid receptors by Holt (2005)10.1038/nmeth778
/ Nat. Methods / A streamlined platform for high-content functional proteomics of primary human specimens by Jessani (2005)10.1038/nm803
/ Nat. Med. / Modulation of anxiety through blockade of anandamide hydrolysis by Kathuria (2003)10.1021/bi002579j
/ Biochemistry / Profiling serine hydrolase activities in complex proteomes by Kidd (2001)10.1016/j.bmcl.2004.12.085
/ Bioorg. Med. Chem. Lett. / Discovery of an exceptionally potent and selective class of fatty acid amide hydrolase inhibitors enlisting proteome-wide selectivity screening: concurrent optimization of enzyme inhibitor potency and selectivity by Leung (2005)10.1038/nbt826
/ Nat. Biotechnol. / Discovering potent and selective reversible inhibitors of enzymes in complex proteomes by Leung (2003)10.1124/jpet.104.069401
/ J. Pharmacol. Exp. Ther. / Reversible inhibitors of fatty acid amide hydrolase that promote analgesia: evidence for an unprecedented combination of potency and selectivity by Lichtman (2004)10.1002/jps.20542
/ J. Pharm. Sci. / Enzymes involved in the bioconversion of ester-based prodrugs by Liederer (2006)10.1074/jbc.M413585200
/ J. Biol. Chem. / Isolation and characterization of a microsomal acid retinyl ester hydrolase by Linke (2005)10.1073/pnas.96.26.14694
/ Proc. Natl. Acad. Sci. U.S.A. / Activity-based protein profiling: the serine hydrolases by Liu (1999)10.1039/b503887a
/ Chem. Commun. (Camb.) / QM/MM modelling of oleamide hydrolysis in fatty acid amide hydrolase (FAAH) reveals a new mechanism of nucleophile activation by Lodola (2005)10.1172/JCI200419465
/ J. Clin. Invest. / The endogenous cannabinoid system protects against colonic inflammation by Massa (2004)10.1146/annurev.biochem.74.082803.133450
/ Annu. Rev. Biochem. / Structure and function of fatty acid amide hydrolase by McKinney (2005)10.1073/pnas.0507470102
/ Proc. Natl. Acad. Sci. U.S.A. / Identification of a high-affinity binding site involved in the transport of endocannabinoids by Moore (2005)10.1021/jm031140x
/ J. Med. Chem. / Cyclohexylcarbamic acid 3′- or 4′-substituted biphenyl-3-yl esters as fatty acid amide hydrolase inhibitors: synthesis, quantitative structure–activity relationships, and molecular modeling studies by Mor (2004)10.1152/ajpheart.00107.2005
/ Am. J. Physiol. Heart Circ. Physiol. / Hemodynamic profile, responsiveness to anandamide, and baroreflex sensitivity of mice lacking fatty acid amide hydrolase by Pacher (2005)10.1002/1615-9861(200109)1:9<1067::AID-PROT1067>3.0.CO;2-4
/ Proteomics / Direct visualization of serine hydrolase activities in complex proteomes using fluorescent active site-directed probes by Patricelli (2001){'key': '10.1016/j.neuropharm.2006.11.009_bib38', 'first-page': '1', 'article-title': 'Involvement of the endogenous cannabinoid system in the effects of alcohol in the mesolimbic reward circuit: electrophysiological evidence in vivo', 'author': 'Perra', 'year': '2005', 'journal-title': 'Psychopharmacology (Berl.)'}
/ Psychopharmacology (Berl.) / Involvement of the endogenous cannabinoid system in the effects of alcohol in the mesolimbic reward circuit: electrophysiological evidence in vivo by Perra (2005){'key': '10.1016/j.neuropharm.2006.11.009_bib39', 'article-title': 'LY2077855: a novel, potent, selective, non-endocannabinoid related inhibitor of anandamide inactivation demonstrates robust analgesic effects in an in vivo pain model', 'author': 'Porter', 'year': '2004', 'journal-title': 'Soc. Neurosci.'}
/ Soc. Neurosci. / LY2077855: a novel, potent, selective, non-endocannabinoid related inhibitor of anandamide inactivation demonstrates robust analgesic effects in an in vivo pain model by Porter (2004)10.1124/jpet.104.081265
/ J. Pharmacol. Exp. Ther. / Hydrolysis of capecitabine to 5′-deoxy-5-fluorocytidine by human carboxylesterases and inhibition by loperamide by Quinney (2005)10.1046/j.1432-1033.2002.03121.x
/ Eur. J. Biochem. / Identification of microsomal rat liver carboxylesterases and their activity with retinyl palmitate by Sanghani (2002)10.1146/annurev.pharmtox.38.1.257
/ Annu. Rev. Pharmacol. Toxicol. / The mammalian carboxylesterases: from molecules to functions by Satoh (1998)- Sit, S.Y., Xie, K., 2002. Bisarylimidazolyl fatty acid amide hydrolase inhibitors. Patent US 6562846 B2.
10.1021/jm049011j
/ J. Med. Chem. / Identification and characterization of novel benzil (diphenylethane-1,2-dione) analogues as inhibitors of mammalian carboxylesterases by Wadkins (2005)10.1124/mol.65.6.1336
/ Mol. Pharmacol. / Discovery of novel selective inhibitors of human intestinal carboxylesterase for the amelioration of irinotecan-induced diarrhea: synthesis, quantitative structure–activity relationship analysis, and biological activity by Wadkins (2004)10.1021/tx015508+
/ Chem. Res. Toxicol. / Synthesis of new carboxylesterase inhibitors and evaluation of potency and water solubility by Wheelock (2001)10.1074/jbc.M511288200
/ J. Biol. Chem. / Association of catsper1 or -2 with Cav3.3 leads to suppression of T-type calcium channel activity by Zhang (2006)
Dates
Type | When |
---|---|
Created | 18 years, 7 months ago (Jan. 10, 2007, 9:28 a.m.) |
Deposited | 6 years, 7 months ago (Jan. 9, 2019, 11:22 p.m.) |
Indexed | 1 year, 1 month ago (July 15, 2024, 1:50 p.m.) |
Issued | 18 years, 6 months ago (March 1, 2007) |
Published | 18 years, 6 months ago (March 1, 2007) |
Published Print | 18 years, 6 months ago (March 1, 2007) |
@article{Zhang_2007, title={Fatty acid amide hydrolase inhibitors display broad selectivity and inhibit multiple carboxylesterases as off-targets}, volume={52}, ISSN={0028-3908}, url={http://dx.doi.org/10.1016/j.neuropharm.2006.11.009}, DOI={10.1016/j.neuropharm.2006.11.009}, number={4}, journal={Neuropharmacology}, publisher={Elsevier BV}, author={Zhang, Di and Saraf, Anita and Kolasa, Teodozyi and Bhatia, Pramila and Zheng, Guo Zhu and Patel, Meena and Lannoye, Greg S. and Richardson, Paul and Stewart, Andrew and Rogers, John C. and Brioni, Jorge D. and Surowy, Carol S.}, year={2007}, month=mar, pages={1095–1105} }