DOI: 10.1016/j.bmcl.2006.03.055. Enhanced pharmacokinetic properties of 1,4-benzodiazepine-2,5-dione antagonists of the HDM2-p53 protein–protein interaction through structure-based drug design

Enhanced pharmacokinetic properties of 1,4-benzodiazepine-2,5-dione antagonists of the HDM2-p53 protein–protein interaction through structure-based drug design

10.1016/j.bmcl.2006.03.055

Crossref journal-article

Elsevier BV

Bioorganic & Medicinal Chemistry Letters (78)

Bibliography

Parks, D. J., LaFrance, L. V., Calvo, R. R., Milkiewicz, K. L., JosÃ© MarugÃ¡n, J., Raboisson, P., Schubert, C., Koblish, H. K., Zhao, S., Franks, C. F., Lattanze, J., Carver, T. E., Cummings, M. D., Maguire, D., Grasberger, B. L., Maroney, A. C., & Lu, T. (2006). Enhanced pharmacokinetic properties of 1,4-benzodiazepine-2,5-dione antagonists of the HDM2-p53 proteinâprotein interaction through structure-based drug design. Bioorganic & Medicinal Chemistry Letters, 16(12), 3310â3314.

Authors 17

Daniel J. Parks (first)
Louis V. LaFrance (additional)
Raul R. Calvo (additional)
Karen L. Milkiewicz (additional)
Juan José Marugán (additional)
Pierre Raboisson (additional)
Carsten Schubert (additional)
Holly K. Koblish (additional)
Shuyuan Zhao (additional)
Carol F. Franks (additional)
Jennifer Lattanze (additional)
Theodore E. Carver (additional)
Maxwell D. Cummings (additional)
Diane Maguire (additional)
Bruce L. Grasberger (additional)
Anna C. Maroney (additional)
Tianbao Lu (additional)

References 14 Referenced 66

10.1038/sj.onc.1208615 / Oncogene by Harris (2005)
10.1158/1535-7163.MCT-04-0327 / Mol. Cancer Ther. by Cao (2005)
10.1158/1541-7786.20.2.1 / Mol. Cancer Res. by Chène (2004)
10.2174/1389557033488178 / Mini-Rev. Med. Chem. by Zheleva (2003)
10.2174/1381612003400911 / Curr. Pharm. Des. by Zhang (2000)
10.1182/blood-2005-02-0553 / Blood by Kojima (2005)
10.4161/cc.3.4.801 / Cell Cycle by Vassilev (2004)
10.1038/sj.bjc.6602164 / Br. J. Cancer by Klein (2004)
10.1126/science.1092472 / Science by Vassilev (2004)
10.1016/j.bmcl.2004.11.009 / Bioorg. Med. Chem. Lett. by Parks (2005)
10.1021/jm049137g / J. Med. Chem. by Grasberger (2005)
10.1158/1535-7163.MCT-05-0199 / Mol. Cancer Ther. by Koblish (2006)
10.1021/jp980230o / J. Phys. Chem. A by Ghose (1998)
10.1016/S0169-409X(00)00129-0 / Adv. Drug Delivery Rev. by Lipinski (2001)

Dates

Type	When
Created	19 years, 4 months ago (April 5, 2006, 11:29 a.m.)
Deposited	2 years, 3 months ago (May 6, 2023, 7:11 p.m.)
Indexed	1 year, 2 months ago (June 8, 2024, 5:53 p.m.)
Issued	19 years, 2 months ago (June 1, 2006)
Published	19 years, 2 months ago (June 1, 2006)
Published Print	19 years, 2 months ago (June 1, 2006)

Funders 0

None

BibTeX

@article{Parks_2006, title={Enhanced pharmacokinetic properties of 1,4-benzodiazepine-2,5-dione antagonists of the HDM2-p53 protein–protein interaction through structure-based drug design}, volume={16}, ISSN={0960-894X}, url={http://dx.doi.org/10.1016/j.bmcl.2006.03.055}, DOI={10.1016/j.bmcl.2006.03.055}, number={12}, journal={Bioorganic & Medicinal Chemistry Letters}, publisher={Elsevier BV}, author={Parks, Daniel J. and LaFrance, Louis V. and Calvo, Raul R. and Milkiewicz, Karen L. and José Marugán, Juan and Raboisson, Pierre and Schubert, Carsten and Koblish, Holly K. and Zhao, Shuyuan and Franks, Carol F. and Lattanze, Jennifer and Carver, Theodore E. and Cummings, Maxwell D. and Maguire, Diane and Grasberger, Bruce L. and Maroney, Anna C. and Lu, Tianbao}, year={2006}, month=jun, pages={3310–3314} }

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