Crossref
journal-article
Elsevier BV
Tetrahedron (78)
References
63
Referenced
44
10.1246/bcsj.73.1053
/ Bull. Chem. Soc. Jpn by Suzuki (2000)-
Watanabe, Y. Angew. Chem. Int. Ed. Engl. 1996, 35, 334-336. (b) Suzuki, M.
(
10.1002/anie.199603341
) - Noyori, R. Chem. Commun. 1999, 307-308. (c) Takechi, H.
-
Watanabe, Y. J. Biol. Chem. 1996, 271, 5901-5906. (d) Satoh, T.
(
10.1074/jbc.271.10.5901
) -
Watanabe, Y. Eur. J. Neurosci. 1999, 11, 3115-3124. (e) Cui, Y.
(
10.1046/j.1460-9568.1999.00791.x
) -
Watanabe, Y. Biochem. Biophys. Res. Commun. 1999, 265, 301-304.
(
10.1006/bbrc.1999.1671
) -
(a) Suzuki, M.; Kato, K.; Noyori, R.; Watanabe, Yu.; Takechi, H.; Matsumura, K.; Långström, B.; Watanabe, Y. Angew. Chem. Int. Ed. Engl. 1996, 35, 334-336.
(
10.1002/anie.199603341
) -
(b) Suzuki, M.; Kato, K.; Watanabe, Yu.; Satoh, T.; Matsumura, K.; Watanabe, Y.; Noyori, R. Chem. Commun. 1999, 307-308.
(
10.1039/a807613h
) -
(c) Takechi, H.; Matsumura, K.; Watanabe, Yu.; Kato, K.; Noyori, R.; Suzuki, M.; Watanabe, Y. J. Biol. Chem. 1996, 271, 5901-5906.
(
10.1074/jbc.271.10.5901
) -
(d) Satoh, T.; Ishikawa, Y.; Kataoka, Y.; Cui, Y.; Yanase, H.; Kato, K.; Watanabe, Yu.; Nakadate, K.; Matsumura, K.; Hatanaka, H.; Kataoka, K.; Noyori, R.; Suzuki, M.; Watanabe, Y. Eur. J. Neurosci. 1999, 11, 3115-3124.
(
10.1046/j.1460-9568.1999.00791.x
) -
(e) Cui, Y.; Kataoka, Y.; Satoh, T.; Yamagata, A.; Shirakawa, N.; Watanabe, Yu.; Suzuki, M.; Yanase, H.; Kataoka, K.; Watanabe, Y. Biochem. Biophys. Res. Commun. 1999, 265, 301-304.
(
10.1006/bbrc.1999.1671
) 10.1046/j.1471-4159.1999.0722583.x
/ J. Neurochem. by Watanabe (1999)10.1016/S1053-8119(97)80002-X
/ NeuroImage by Watanabe (1997)10.3891/acta.chem.scand.52-0635
/ Acta Chem. Scand. by Björkman (1998)10.1002/chem.19970031219
/ Chem. Eur. J. by Suzuki (1997)-
For the Stille reaction, see: (a) Stille, J. K. Angew. Chem. Int. Ed. Engl. 1986, 25, 508-524.
(
10.1002/anie.198605081
) -
Groh, B. L. J. Am. Chem. Soc. 1987, 109, 813-817. (c) Farina, V.
(
10.1021/ja00237a029
) -
Scott, W. J. Org. React. 1997, 50, 1-652. (d) Motchell, T. N. Synthesis 1992, 803-815. (e) Farina, V. Pure Appl. Chem. 1996, 68, 73-78. (f) Farina, V.
(
10.1351/pac199668010073
) -
(a) Stille, J. K. Angew. Chem. Int. Ed. Engl. 1986, 25, 508-524.
(
10.1002/anie.198605081
) -
(b) Stille, J. K.; Groh, B. L. J. Am. Chem. Soc. 1987, 109, 813-817.
(
10.1021/ja00237a029
) -
(c) Farina, V.; Krishnamurthy, V.; Scott, W. J. Org. React. 1997, 50, 1-652.
(
10.1002/0471264180.or050.01
) -
(d) Motchell, T. N. Synthesis 1992, 803-815.
(
10.1055/s-1992-26230
) -
(e) Farina, V. Pure Appl. Chem. 1996, 68, 73-78.
(
10.1351/pac199668010073
) - (f) Farina, V.; Roth, G. P. In Advances in Metal-Organic Chemistry; Liebeskind, L. S., Ed.; JAI Press: 1996; Vol. 5, pp 1-53.
-
Chapters 9-11. (b) Fowler, J. S., Wolf, A. P. Acc. Chem. Res. 1997, 30, 181-188. (c) Långström, B.
(
10.1021/ar960068c
) - W. B. Saunders: Philadelphia, 1995
-
Section 1, Chapter 11. (d) Brennan, M. B. Chem. Eng. News 1996, 74 (Feb. 19), pp 26-33 (e) Långström, B.
(
10.1021/cen-v074n008.p026
) -
Ögren, M. Acta Chem. Scand. 1999, 53, 651-669.
(
10.3891/acta.chem.scand.53-0651
) - (a) Fowler, J. S.; Wolf, A. P.; Barrio, J. R.; Mazziotta, J. C.; Phelps, M. E. In Positron Emission Tomography and Autoradiography; Phelps, M. E., Mazziotta, J. C., Schelbert, H. R., Eds.; Raven Press: New York, 1986; Chapters 9-11.
-
(b) Fowler, J. S., Wolf, A. P. Acc. Chem. Res. 1997, 30, 181-188.
(
10.1021/ar960068c
) - (c) Långström, B.; Dannals, R. F. In Principles of Nuclear Medicine, 2nd ed.; Wagner, H. N., Szabo, Z., Buchanan. J. W., Eds.; W. B. Saunders: Philadelphia, 1995; Section 1, Chapter 11.
-
(d) Brennan, M. B. Chem. Eng. News 1996, 74 (Feb. 19), pp 26-33
(
10.1021/cen-v074n008.p026
) -
(e) Långström, B.; Kihlberg, T.; Bergström, M.; Antoni, G.; Björkman, M.; Forngren, B. H.; Forngren, T.; Hartvig, P.; Markides, K.; Yngve, U.; Ögren, M. Acta Chem. Scand. 1999, 53, 651-669.
(
10.3891/acta.chem.scand.53-0651
) - The methyl ester [11C]-6 was assumed to penetrate the blood–brain-barrier (BBB) and then to be hydrolyzed to be the corresponding acid form [11C]-5 which binds to the receptor in the brain. See references 1 and 4.
-
Svärd, H. J. Nucl. Med. 1987, 28, 1037-1040. (b) Ferrieri, R. A.
(
10.1016/0032-3861(87)90182-0
) -
Wolf, A. P. Radiochim. Acta 1983, 34, 69-83.
(
10.1016/S0020-1693(00)83555-0
) - (a) Långström, B.; Antoni, G.; Gullberg, P.; Halldin, C.; Malmborg, P.; Någren, K.; Rimland, A.; Svärd, H. J. Nucl. Med. 1987, 28, 1037-1040.
-
(b) Ferrieri, R. A.; Wolf, A. P. Radiochim. Acta 1983, 34, 69-83.
(
10.1524/ract.1983.34.12.69
) - The methylation with stannyl precursors, 7 and 10, under the conditions used in entry 5 in Table 1 (one-pot operation) gave 15R-TIC methyl ester [12C]-6 and 15-deoxy-TIC methyl ester [12C]-11 in 82 and 92% yield, respectively.
- Details will be reported separately.
- The investigation for healthy volunteers and patients is in progress. Recently, the principal author (M. S.) chosen as a first volunteer succeeded in imaging the IP2 receptor in his brain.
-
Migita, T. Bull. Chem. Soc. Jpn 1983, 56, 3855-3856. (b) Kosugi, M.
(
10.1246/bcsj.56.3855
) -
Migita T. Chem. Lett. 1981, 829-830.
(
10.1055/s-1981-29617
) -
(a) Kosugi, M.; Ohya, T.; Migita, T. Bull. Chem. Soc. Jpn 1983, 56, 3855-3856.
(
10.1246/bcsj.56.3855
) -
(b) Kosugi, M.; Shimizu, K.; Ohtani, A.; Migita T. Chem. Lett. 1981, 829-830.
(
10.1246/cl.1981.829
) -
Noyori, R. Tetrahedron 1992, 48, 2635-2658. (b) Sodeoka, M.
(
10.1016/S0040-4020(01)88526-4
) -
Shibasaki, M. Chem. Pharm. Bull. 1989, 37, 586-598. (c) Hemmerle, H.
(
10.1248/cpb.37.586
) -
Gais, H.-J. Angew. Chem. Int. Ed. Engl. 1989, 28, 349-351. (d) Manabe, K.
(
10.1002/anie.198903491
) -
Kato, Y. J. Labelled Compds. Radiopharm. 1991, 29, 1107-1119.
(
10.1002/jlcr.2580291003
) -
(a) Suzuki, M.; Koyano, H.; Noyori, R. Tetrahedron 1992, 48, 2635-2658.
(
10.1016/S0040-4020(01)88526-4
) -
(b) Sodeoka, M.; Ogawa, Y.; Mase, T.; Shibasaki, M. Chem. Pharm. Bull. 1989, 37, 586-598.
(
10.1248/cpb.37.586
) -
(c) Hemmerle, H.; Gais, H.-J. Angew. Chem. Int. Ed. Engl. 1989, 28, 349-351.
(
10.1002/anie.198903491
) -
(d) Manabe, K.; Tanaka, T.; Kurozumi, S.; Kato, Y. J. Labelled Compds. Radiopharm. 1991, 29, 1107-1119.
(
10.1002/jlcr.2580291003
) -
(a) Luche, J.-L. J. Am. Chem. Soc. 1978, 100, 2226-2227. (b) Luche, J.-L.
(
10.1021/ja00475a040
) - Crabbé, P. J. Chem. Soc., Chem. Commun. 1978, 601-602.
-
(a) Luche, J.-L. J. Am. Chem. Soc. 1978, 100, 2226-2227.
(
10.1021/ja00475a040
) -
(b) Luche, J.-L.; Rodriguez-Hahn, L.; Crabbé, P. J. Chem. Soc., Chem. Commun. 1978, 601-602.
(
10.1039/C39780000601
) 10.1039/jr9610001266
/ J. Chem. Soc. by Trippett (1961)-
Minami, I. Acc. Chem. Res. 1987, 20, 140-145. (b) Tsuji, J. Tetrahedron 1986, 42, 4361-4401. (c) Tsuji, J.
(
10.1016/S0040-4020(01)87277-X
) -
Takahashi, K. J. Org. Chem. 1985, 50, 1523-1529.
(
10.1021/jo00209a032
) -
(a) Tsuji, J.; Minami, I. Acc. Chem. Res. 1987, 20, 140-145.
(
10.1021/ar00136a003
) -
(b) Tsuji, J. Tetrahedron 1986, 42, 4361-4401.
(
10.1016/S0040-4020(01)87277-X
) -
(c) Tsuji, J.; Shimizu, I.; Minami, I.; Ohashi, Y.; Sugiura, T.; Takahashi, K. J. Org. Chem. 1985, 50, 1523-1529.
(
10.1021/jo00209a032
)
Dates
Type | When |
---|---|
Created | 23 years, 1 month ago (July 25, 2002, 10:41 a.m.) |
Deposited | 3 years, 2 months ago (June 24, 2022, 6:54 p.m.) |
Indexed | 6 months, 1 week ago (Feb. 20, 2025, 11:34 p.m.) |
Issued | 24 years, 11 months ago (Oct. 1, 2000) |
Published | 24 years, 11 months ago (Oct. 1, 2000) |
Published Print | 24 years, 11 months ago (Oct. 1, 2000) |
Funders
1
Ministry of Education, Culture, Sports, Science and Technology
10.13039/501100001700
Region: Asia
gov (National government)
Labels
3
- Monbu-kagaku-shō
- 文部科学省
- MEXT
@article{Suzuki_2000, title={Rapid Methylation for the Synthesis of a 11C-Labeled Tolylisocarbacyclin Imaging the IP2 Receptor in a Living Human Brain}, volume={56}, ISSN={0040-4020}, url={http://dx.doi.org/10.1016/s0040-4020(00)00734-1}, DOI={10.1016/s0040-4020(00)00734-1}, number={42}, journal={Tetrahedron}, publisher={Elsevier BV}, author={Suzuki, Masaaki and Doi, Hisashi and Kato, Koichi and Björkman, Margareta and Långström, Bengt and Watanabe, Yasuyoshi and Noyori, Ryoji}, year={2000}, month=oct, pages={8263–8273} }