DOI: 10.1016/0145-2126(86)90050-0. An inhibitor of protein kinase C, 1-(5-isoquinolinylsulfonyl)-2-methylpiperazine(H-7) inhibits TPA-induced reduction of vincristine uptake from P388 murine leukemic cell

An inhibitor of protein kinase C, 1-(5-isoquinolinylsulfonyl)-2-methylpiperazine(H-7) inhibits TPA-induced reduction of vincristine uptake from P388 murine leukemic cell

10.1016/0145-2126(86)90050-0

Crossref journal-article

Elsevier BV

Leukemia Research (78)

Bibliography

Ido, M., Asao, T., Sakurai, M., Inagaki, M., Saito, M., & Hidaka, H. (1986). An inhibitor of protein kinase C, 1-(5-isoquinolinylsulfonyl)-2-methylpiperazine(H-7) inhibits TPA-induced reduction of vincristine uptake from P388 murine leukemic cell. Leukemia Research, 10(9), 1063â1069.

Authors 6

Masaru Ido (first)
Toyohiko Asao (additional)
Minoru Sakurai (additional)
Masaki Inagaki (additional)
Masahiro Saito (additional)
Hiroyoshi Hidaka (additional)

References 23 Referenced 32

{'key': '10.1016/0145-2126(86)90050-0_BIB1', 'first-page': '1967', 'article-title': 'Overcoming of vincristine resistance in P388 leukemia in vivo and in vitro through enhanced cytotoxicity of vincristine and vinblastine by verapamil', 'volume': '41', 'author': 'Tsuruo', 'year': '1981', 'journal-title': 'Cancer Res.'} / Cancer Res. / Overcoming of vincristine resistance in P388 leukemia in vivo and in vitro through enhanced cytotoxicity of vincristine and vinblastine by verapamil by Tsuruo (1981)
{'key': '10.1016/0145-2126(86)90050-0_BIB2', 'first-page': '4730', 'article-title': 'Increased accumulation of vincristine and adriamycin in drug-resistant P388 tumor cells following incubation with calcium antagonists and calmodulin inhibitors', 'volume': '42', 'author': 'Tsuruo', 'year': '1982', 'journal-title': 'Cancer Res.'} / Cancer Res. / Increased accumulation of vincristine and adriamycin in drug-resistant P388 tumor cells following incubation with calcium antagonists and calmodulin inhibitors by Tsuruo (1982)
{'key': '10.1016/0145-2126(86)90050-0_BIB3', 'first-page': '1687', 'article-title': 'Anthracycline resistance in P388 murine leukemia and its circumvention by calcium antagonists', 'volume': '45', 'author': 'Kessel', 'year': '1985', 'journal-title': 'Cancer Res.'} / Cancer Res. / Anthracycline resistance in P388 murine leukemia and its circumvention by calcium antagonists by Kessel (1985)
{'key': '10.1016/0145-2126(86)90050-0_BIB4', 'first-page': '1651', 'article-title': 'Verapamil-induced augmentation of etoposide accumulation in L1210 cells in vitro', 'volume': '45', 'author': 'Yalowich', 'year': '1985', 'journal-title': 'Cancer Res.'} / Cancer Res. / Verapamil-induced augmentation of etoposide accumulation in L1210 cells in vitro by Yalowich (1985)
10.1016/S0021-9258(17)41009-X / J. biol. Chem. / Studies on cyclic nucleotide-independent protein kinase and its proenzyme in mammalian tissues by Takai (1977)
10.1016/0024-3205(81)90026-6 / Life Sci. / Inhibition by phenothiazine antipsychotic drugs of calcium-dependent phosphorylation of cerebral cortex proteins regulated by phospholipid or calmodulin by Wrenn (1981)
Wise B.C. & Kuo J.F. Modes of inhibition by acylcarnitines, adriamycin, and trifluoperazine of cardiac phospholipid-sensitive calcium-dependent protein kinase. Biochem. Pharmac.32, 1259. (10.1016/0006-2952(83)90280-0)
{'key': '10.1016/0145-2126(86)90050-0_BIB8', 'first-page': '7039', 'article-title': 'Calcium-dependent protein kinase: widespread occurrence in various tissues and phyla of the animal kingdom and comparison of effects of phospholipid, calmodulin, and trifluoperazine', 'volume': '77', 'author': 'Kuo', 'year': '1980'} / Calcium-dependent protein kinase: widespread occurrence in various tissues and phyla of the animal kingdom and comparison of effects of phospholipid, calmodulin, and trifluoperazine by Kuo (1980)
10.1038/308693a0 / Nature, Lond. / The role of protein kinase C in cell surface signal transduction and tumor promotion by Nishizuka (1984)
{'key': '10.1016/0145-2126(86)90050-0_BIB10', 'first-page': '36', 'article-title': 'Phorbol diester receptor copurifies with protein kinase C', 'volume': '80', 'author': 'Niedel', 'year': '1983'} / Phorbol diester receptor copurifies with protein kinase C by Niedel (1983)
{'key': '10.1016/0145-2126(86)90050-0_BIB11', 'first-page': '2955', 'article-title': 'Phospholipid-sensitive Ca2+-dependent protein phosphorylation system in various types of leukemic cells from human patients and in human leukemic cell lines HL60 and K562, and its inhibition by alkyl-lysophospholipid', 'volume': '43', 'author': 'Helfman', 'year': '1983', 'journal-title': 'Cancer Res.'} / Cancer Res. / Phospholipid-sensitive Ca2+-dependent protein phosphorylation system in various types of leukemic cells from human patients and in human leukemic cell lines HL60 and K562, and its inhibition by alkyl-lysophospholipid by Helfman (1983)
10.1021/bi00316a032 / Biochemistry / Isoquinolinesulfonamides, novel and potent inhibitors of cyclic nucleotide dependent protein kinase and protein kinase C by Hidaka (1984)
{'key': '10.1016/0145-2126(86)90050-0_BIB13', 'first-page': '1521', 'article-title': 'Resistance and cross-resistance of cultured leukemia P388 cells to vincristine, adriamycin, adriamycin analogs and actinomycin D', 'volume': '61', 'author': 'Wilkoff', 'year': '1978', 'journal-title': 'J. natn. Cancer Inc.'} / J. natn. Cancer Inc. / Resistance and cross-resistance of cultured leukemia P388 cells to vincristine, adriamycin, adriamycin analogs and actinomycin D by Wilkoff (1978)
{'key': '10.1016/0145-2126(86)90050-0_BIB14', 'first-page': '1189', 'article-title': 'Specific receptors for phorbol esters in lymphoid cell populations: role in enhanced production of T-cell growth factor', 'volume': '78', 'author': 'Sando', 'year': '1981'} / Specific receptors for phorbol esters in lymphoid cell populations: role in enhanced production of T-cell growth factor by Sando (1981)
10.1016/S0021-9258(18)89453-4 / J. biol. Chem. / N-(2-aminoethyl)-5-isoquinolinesulfonamide, a newly synthesized protein kinase inhibitor functions as a ligand in affinity chromatography; purification of Ca2+-activated, phospholipid dependent and other protein kinases by Inagaki (1985)
Schulman H. in Handbook of Experimental Pharmacology 58/I (Nathason, J. A. & Kebabian, J. W., Eds.), p. 425. Springer, New York.
10.1016/S0021-9258(18)33453-7 / J. biol. Chem. / Calcium-activated, phospholipid-dependent protein kinase from rat brain by Kikkawa (1982)
10.1042/bj2090435 / Biochem. J. / Purification to homogeneity, characterization and monoclonal antibodies of phospholipid-sensitive Ca2+-dependent protein kinase from spleen by Schatzman (1983)
10.1042/bj2240483 / Biochem. J. / Phorbol ester stimulation of insulin release and secretory-granule protein phosphorylation in a transplantable rat insulinoma by Hutton (1984)
10.1016/S0021-9258(17)42594-4 / J. biol. Chem. / Serotonin secretion from human platelets may be modified by Ca2+-activated phospholipid-dependent myosin phosphorylation by Inagaki (1984)
{'key': '10.1016/0145-2126(86)90050-0_BIB21', 'first-page': '63', 'article-title': 'Uptake of adriamycin and daunomycin in L1210 and human leukemic cells: A comparative study', 'volume': '7', 'author': 'Chervinsky', 'year': '1976', 'journal-title': 'J. Med.'} / J. Med. / Uptake of adriamycin and daunomycin in L1210 and human leukemic cells: A comparative study by Chervinsky (1976)
10.1016/0005-2736(73)90191-0 / Biochim. Biophys. Acta / Active outward transport of daunomycin in resistant Ehrlich ascites tumor cells by Danø (1973)
{'key': '10.1016/0145-2126(86)90050-0_BIB23', 'first-page': '4722', 'article-title': 'Mechanism of cross-resistance between vincristine and daunomycin in Ehrlich ascites tumor cells', 'volume': '38', 'author': 'Skovsgaard', 'year': '1978', 'journal-title': 'Cancer Res.'} / Cancer Res. / Mechanism of cross-resistance between vincristine and daunomycin in Ehrlich ascites tumor cells by Skovsgaard (1978)

Dates

Type	When
Created	21 years, 4 months ago (April 19, 2004, 9:46 a.m.)
Deposited	4 years, 2 months ago (June 16, 2021, 3:28 a.m.)
Indexed	1 month, 2 weeks ago (July 14, 2025, 11:43 p.m.)
Issued	39 years, 8 months ago (Jan. 1, 1986)
Published	39 years, 8 months ago (Jan. 1, 1986)
Published Print	39 years, 8 months ago (Jan. 1, 1986)

Funders 0

None

BibTeX

@article{Ido_1986, title={An inhibitor of protein kinase C, 1-(5-isoquinolinylsulfonyl)-2-methylpiperazine(H-7) inhibits TPA-induced reduction of vincristine uptake from P388 murine leukemic cell}, volume={10}, ISSN={0145-2126}, url={http://dx.doi.org/10.1016/0145-2126(86)90050-0}, DOI={10.1016/0145-2126(86)90050-0}, number={9}, journal={Leukemia Research}, publisher={Elsevier BV}, author={Ido, Masaru and Asao, Toyohiko and Sakurai, Minoru and Inagaki, Masaki and Saito, Masahiro and Hidaka, Hiroyoshi}, year={1986}, month=jan, pages={1063–1069} }

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